About 24 results.

Metitepine

Description. Lang: en

Metitepine (INN; developmental code names Ro 8-6837 (maleate), VUFB-6276 (mesylate)), also known as methiothepin, is a drug described as a "psychotropic agent" of the tricyclic group which was never marketed. It acts as a non-selective antagonist of serotonin, dopamine, and adrenergic receptors and has antipsychotic properties.
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Metitepine

Metitepine

Drug

  • Desc: Metitepine, also known as methiothepin, is a drug described as a "psychotropic agent" of the tricyclic group which was never marketed. It acts as a non-selective antagonist of serotonin, dopamine, and adrenergic receptors and has antipsychotic properties.
  • Wiki: https://en.wikipedia.org/wiki/Metitepine
  • Type: Thing
  • Result Score: 34.70
Methamnetamine

Methamnetamine

Drug

  • Desc: Methamnetamine is a triple monoamine releasing agent and N-methyl analog of the non-neurotoxic experimental drug naphthylaminopropane and the naphthalene analog of methamphetamine. It has been sold online as a designer drug.
  • Wiki: https://en.wikipedia.org/wiki/Methamnetamine
  • Type: Thing
  • Result Score: 6.47

PRX-03140

Pharmaceutical

  • Desc: PRX-03140 is a partial agonist of the 5-HT₄ receptor that is being developed by EPIX Pharmaceuticals for Alzheimer's disease.
  • Wiki: https://en.wikipedia.org/wiki/PRX-03140
  • Type: Thing
  • Result Score: 6.33
Roluperidone

Roluperidone

Drug

  • Desc: Roluperidone is a 5-HT2A and σ₂ receptor antagonist that is under development by Minerva Neurosciences for the treatment of schizophrenia. One of its metabolites also has some affinity for the H₁ receptor. As of May 2018, the drug is in phase III clinical trials.
  • Wiki: https://en.wikipedia.org/wiki/Roluperidone
  • Type: Thing
  • Result Score: 6.24
Perathiepin

Perathiepin

Drug

  • Desc: Perathiepin is a neuroleptic drug of the tricyclic family which was developed in the 1960s but was never marketed. In animal studies it was found to possess central depressant, antihistamine, antiserotonergic, and analgesic effects.
  • Wiki: https://en.wikipedia.org/wiki/Perathiepin
  • Type: Thing
  • Result Score: 5.57

Aripiprazole/sertraline

Pharmaceutical

  • Desc: Aripiprazole/sertraline is a combination formulation of sertraline, a selective serotonin reuptake inhibitor, and aripiprazole, an atypical antipsychotic, which is under development by Otsuka Pharmaceutical for the treatment of major depressive disorder.
  • Wiki: https://en.wikipedia.org/wiki/Aripiprazole/sertraline
  • Type: Thing
  • Result Score: 5.56

AVN-101

Pharmaceutical

  • Desc: AVN-101, a close structural analogue of latrepirdine, is a selective 5-HT₆ receptor antagonist which is under development by Avineuro Pharmaceuticals for the treatment of Alzheimer's disease and anxiety disorders.
  • Wiki: https://en.wikipedia.org/wiki/AVN-101
  • Type: Thing
  • Result Score: 5.36
N-Feruloylserotonin

N-Feruloylserotonin

Chemical compound

  • Desc: N-Feruloylserotonin an alkaloid and polyphenol found in safflower seed. Chemically, it is an amide formed between serotonin and ferulic acid. It has in vitro anti-atherogenic activity.
  • Wiki: https://en.wikipedia.org/wiki/N-Feruloylserotonin
  • Type: Thing
  • Result Score: 5.20
Promazine

Promazine

Medication

  • Desc: Promazine is a medication that belongs to the phenothiazine class of antipsychotics. An older medication used to treat schizophrenia, it is still prescribed, alongside newer agents such as olanzapine and quetiapine.
  • Wiki: https://en.wikipedia.org/wiki/Promazine
  • Type: Thing
  • Result Score: 5.16
LY-215,840

LY-215,840

Drug

  • Desc: LY-215,840 is an ergoline derivative drug developed by Eli Lilly, which acts as a potent and selective antagonist at the serotonin 5-HT₂ and 5-HT₇ receptors. It has anti-hypertensive and muscle relaxant effects in animal studies.
  • Wiki: https://en.wikipedia.org/wiki/LY-215,840
  • Type: Thing
  • Result Score: 5.11
Urapidil

Urapidil

Drug

  • Desc: Urapidil is a sympatholytic antihypertensive drug. It acts as an α₁-adrenoceptor antagonist and as an 5-HT1A receptor agonist. Although an initial report suggested that urapidil was also an α₂-adrenoceptor agonist, this was not substantiated in later studies that demonstrated it was devoid of agonist actions in the dog saphenous vein and the guinea-pig ileum.
  • Wiki: https://en.wikipedia.org/wiki/Urapidil
  • Type: Thing
  • Result Score: 5.07
NM-2-AI

NM-2-AI

Drug

  • Desc: NM-2-AI is a psychoactive drug and research chemical that has been sold online as a designer drug. It is a rigid analogue of methamphetamine. It is a derivative of 2-aminoindane.
  • Wiki: https://en.wikipedia.org/wiki/NM-2-AI
  • Type: Thing
  • Result Score: 4.97
Metergoline

Metergoline

Drug

  • Desc: Metergoline is a psychoactive drug of the ergoline chemical class which acts as a ligand for various serotonin and dopamine receptors.
  • Wiki: https://en.wikipedia.org/wiki/Metergoline
  • Type: Thing
  • Result Score: 4.96
Cyamemazine

Cyamemazine

Drug

  • Desc: Cyamemazine, also known as cyamepromazine, is a typical antipsychotic drug of the phenothiazine class which was introduced by Theraplix in France in 1972 and later in Portugal as well.
  • Wiki: https://en.wikipedia.org/wiki/Cyamemazine
  • Type: Thing
  • Result Score: 4.96

Opiranserin

Drug

  • Desc: Opiranserin is a selective and combined glycine GlyT2 transporter blocker, purine P2X₃ receptor antagonist, and serotonin 5-HT2A receptor antagonist which is under development by Vivozon for the intravenous treatment of postoperative pain.
  • Wiki: https://en.wikipedia.org/wiki/Opiranserin
  • Type: Thing
  • Result Score: 4.96
Eltoprazine

Eltoprazine

Drug

  • Desc: Eltoprazine is a drug of the phenylpiperazine class which is a serenic or antiaggressive agent. It acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.
  • Wiki: https://en.wikipedia.org/wiki/Eltoprazine
  • Type: Thing
  • Result Score: 4.76
Iferanserin

Iferanserin

Drug

  • Desc: Iferanserin is a drug which acts as a selective 5-HT2A receptor antagonist. It is under development as an intra-rectal formulation for the treatment of hemorrhoid disease, and as of February 2012, is in phase IIb clinical trials.
  • Wiki: https://en.wikipedia.org/wiki/Iferanserin
  • Type: Thing
  • Result Score: 4.73
Elopiprazole

Elopiprazole

Drug

Tranylcypromine/trifluoperazine

Drug

  • Desc: Tranylcypromine/trifluoperazine is a combination formulation of the monoamine oxidase inhibitor antidepressant drug tranylcypromine and the typical antipsychotic drug trifluoperazine that has been used in the treatment of major depressive disorder.
  • Wiki: https://en.wikipedia.org/wiki/Tranylcypromine/trifluoperazine
  • Type: Thing
  • Result Score: 4.51
Quipazine

Quipazine

Drug

  • Desc: Quipazine is a piperazine drug used in scientific research. It is a moderately selective serotonin receptor receptor agonist, binding to a range of different serotonin receptors, but particularly to the 5-HT2A and 5-HT₃.
  • Wiki: https://en.wikipedia.org/wiki/Quipazine
  • Type: Thing
  • Result Score: 4.48
Melitracen

Melitracen

Drug

  • Desc: Melitracen is a tricyclic antidepressant marketed in Europe and Japan by Lundbeck and Takeda, respectively, for the treatment of depression and anxiety.
  • Wiki: https://en.wikipedia.org/wiki/Melitracen
  • Type: Thing
  • Result Score: 4.47
LY-310762

LY-310762

Drug

  • Desc: LY-310762 is a drug which acts as a potent and selective antagonist for the 5-HT1D serotonin receptor, with reasonable selectivity over the closely related 5-HT1B subtype.
  • Wiki: https://en.wikipedia.org/wiki/LY-310762
  • Type: Thing
  • Result Score: 4.45
SB-206553

SB-206553

Drug

  • Desc: SB-206553 is a drug which acts as a mixed antagonist for the 5-HT2B and 5-HT2C serotonin receptors. It has anxiolytic properties in animal studies and interacts with a range of other drugs.
  • Wiki: https://en.wikipedia.org/wiki/SB-206553
  • Type: Thing
  • Result Score: 4.40
Tolpiprazole

Tolpiprazole

Drug

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